理化学研究所 ライフサイエンス技術基盤研究センター
分子標的化学研究チーム
RIKEN Center for Life Science Technologies (CLST)
Chemical Biology Team
論 文 リ ス ト （2016年6月現在）
隅田 有人
Original papers:
18.
Preparation of Aryne−Nickel Complexes from ortho-Borylaryl Triflates
Yuto Sumida, Tomoe Sumida, Daisuke Hashizume, Takamitsu Hosoya*,
Org. Lett. 2016, 18, 5600–5603.
DOI: 10.1021/acs.orglett.6b02831
17.
Selective inhibition of the kinase DYRK1A by targeting its folding process
I. Kii*, Y. Sumida, T. Goto, R. Sonamoto, Y Okuno, S. Yoshida, T. Kato-Sumida, Y. Koike, M. Abe, Y. Nonaka, T. Ikura, N. Ito, H. Shibuya, T. Hosoya, M. Hagiwara*,
Nat. Commun. 2016, 7, 11391.
DOI: 10.1038/ncomms11391
16.
Concise Synthesis of v-Coelenterazines
T. Hosoya*, R. Iimori, S. Yoshida, Y. Sumida, Y. Sahara-Miura, J.-i. Sato, S. Inouye,
Org. Lett. 2015, 17, 3888–3891.
DOI: 10.1021/acs.orglett.5b01872
15.
Identification of a DYRK1A Inhibitor that Induces Degradation of the Target Kinase using
Co-chaperone CDC37 fused with Luciferase nanoKAZ
R. Sonamoto, I. Kii, Y. Koike, Y. Sumida, T. Kato-Sumida, T. Hosoya, M. Hagiwara*
Sci. Rep. 2015, 5, 12728.
14.
Design and synthesis of a potent inhibitor of class 1 DYRK kinases as a suppressor of adipogenesis
S. Masaki, I. Kii, Y. Sumida, T. Kato-Sumida Y. Ogawa, N. Ito, M. Nakamura, R. Sonamoto, N. Kataoka, T. Hosoya, M. Hagiwara*
Bioorg. Med. Chem. 2015, 23, 4434–4441.
13.
An Alternative Method for Generating Arynes from ortho-Silylaryl Triflates: Activation by Cesium
Carbonate in the Presence of a Crown Ether
S. Yoshida, Y. Hazama, Y. Sumida, T. Yano, T. Hosoya*
Molecules 2015, 20, 10131–10140.
DOI:10.3390/molecules200610131
12.
Boron-Selective Biaryl Coupling Approach to Versatile Dibenzoxaborins and Application to Concise Synthesis of Defucogilvocarcin M.
Y. Sumida, R. Harada, T. Kato-Sumida, K. Johmoto, H. Uekusa, *T. Hosoya.
Org. Lett. 2014, 16, 6240–6243.
11.
Generation of Arynes via Ate Complexes of Arylboronic Esters with an ortho-Leaving Group.
Y. Sumida, T. Kato, *T. Hosoya.
Org. Lett. 2013, 15, 2806–2809.
10.
Palladium-Catalyzed Regio- and Stereoselective Hydrosilylation of Electron-Deficient Alkynes.
*Y. Sumida, T. Kato, S. Yoshida, *T. Hosoya.
Org. Lett. 2012, 14, 1552–1555.
9.
Primer Preactivation of Peptidoglycan Polymerases.
T-S. A. Wang, T. J. Lupoli, Y. Sumida, H. Tsukamoto, Y. Wu, Y. Rebets, D. E. Kahne, *S. Walker.
J. Am. Chem. Soc. 2011, 133, 8528–8530.
8.
Nickel-Catalyzed Arylative Ring-Opening of 3-Methylenecycloalkane-1,1- dicarboxylate.
Y. Sumida, *H. Yorimitsu, *K. Oshima.
Org. Lett. 2010, 12, 2254–2257.
7.
Radical Addition of Polyhaloalkanes to 2-Ethynyl-4,4,5,5-tetramethyl-1,3-2-dioxaboronate.
T. Wada, Y. Sumida, A. Kondoh, *H. Yorimitsu, *K. Oshima.
Bull. Chem. Soc. Jpn. 2009, 82, 1433–1435.
6.
Palladium-Catalyzed Preparation of Silyl Enolates from α,β-Unsaturated Ketones or Cyclopropyl Ketones with Hydrosilanes.
Y. Sumida, *H. Yorimitsu, *K. Oshima.
J. Org. Chem. 2009, 74, 7986–7989.
5.
Nickel-Catalyzed Borylation of Aryl Cyclopropyl Ketones with Bis(pinacolato)diboron to Synthesize 4-Oxoalkylboronates.
Y. Sumida, *H. Yorimitsu, *K. Oshima.
J. Org. Chem. 2009, 74, 3196–3198.
4.
Nickel-Catalyzed Borylative Ring-Opening Reaction of Vinylcyclopropanes with Bis(pinacolato)diboron Yielding Allylic boronates.
Y. Sumida, *H. Yorimitsu, *K. Oshima.
Org. Lett. 2008, 10, 4677–4679.
3.
Nickel-Catalyzed Allylation of Allyl Carbonates with Homoallyl Alcohols via
Retro-Allylation Providing 1,5-Hexadienes.
Y. Sumida, S. Hayashi, K. Hirano, *H. Yorimitsu, *K. Oshima.
Org. Lett. 2008, 10, 1629–1632.
2.
Rhodium-Catalyzed Allylation of Aldehydes with Homoallyl Alcohols via Retroallylation and Isomerization to Saturated Ketones with Conventional or Microwave Heating.
Y. Sumida, Y. Takada, S. Hayashi, K. Hirano, *H. Yorimitsu, *K. Oshima.
Chem. Asian J. 2008, 1, 119–125.
1.
Discrepancy of the spectral data between adunctin E and the synthetic one,
*M. Yamashita, N. D. Yadav, Y. Sumida, I. Kawasaki, A. Kurume, *S. Ohta.
Tetrahedron Lett. 2007, 48, 5619–5622.
DOI:10.1016/j.tetlet.2007.06.050
